Valemetostat (DS-3201) is a First-in-class EZH1/2 Dual Inhibitor for Adult T-cell Leukemia Research
Enhancer of zeste homolog 2 (EZH2) is a histone-lysine N-methyltransferase enzyme encoded by EZH2 gene. And it participates in histone methylation and, ultimately, transcriptional repression. Meanwhile, mutation or over-expression of…