BI-9321, a First-in-Class Chemical Probe, is a NSD3-PWWP1 Inhibitor
Post-translational modification of histones by histone-modifying enzymes represents a key element of epigenetic regulation. Epigenetic reader domains are structurally diverse. They include bromodomains, PHD domains, methyl-lysine- and/or methyl-arginine-binding domains, frequently…