BAY-8002, a Monocarboxylate Transporter 1 Inhibitor for Cancer Research
MCTs (Monocarboxylate Transporters) are proton coupled monocarboxylate transporter. They can carry lactate and pyruvate across biological membranes. MCT1, also called SLC16A1, has a vital role in tumor cell energy homeostasis. Inhibition of lactate transport has effects on tumor growth. Cancer cells accumulate intracellular lactate if the lactate transport is...